SCHEMBL290106

SCHEMBL290106

COCCn1c(=O)oc2ccc(-c3ccc(CCN(C#N)C(=O)C4(NC(=O)O)CCOCC4)cc3)cc21

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSC P53634 8/20 0.46
TSPO P30536 1/20 0.36
KCNH2 Q12809 1/20 0.35
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ASAH1 Q13510 1/20 0.34
KMO O15229 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290462 0.96 CTSC (0.46) CTSCTSPOKCNH2ASAH1
SCHEMBL290319 0.89 CTSC (0.42) CTSCKCNH2ASAH1
SCHEMBL290292 0.86 CTSC (0.47) CTSCKCNH2
SCHEMBL2890775 0.82 CTSC (0.62) CTSCKCNH2
SCHEMBL290107 0.80 CTSC (0.49) CTSCTSPOKCNH2KMO
SCHEMBL290245 0.79 CTSS (0.39) POLBL3MBTL1
SCHEMBL299685 0.78 CTSC (0.49) CTSCKCNH2
SCHEMBL288780 0.78 CTSC (0.40) CTSC
SCHEMBL2885392 0.78 CTSC (0.62) CTSCKCNH2
SCHEMBL289727 0.76 CTSC (0.54) CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed