SCHEMBL290292

SCHEMBL290292

COCCn1c(=O)sc2ccc(-c3ccc(CCN(C#N)C(=O)C4(NC(=O)O)CCOCC4)cc3)cc21

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSC P53634 5/20 0.47
KCNH2 Q12809 1/20 0.35
CTSK P43235 1/20 0.31
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290106 0.86 CTSC (0.46) CTSCKCNH2
SCHEMBL290462 0.82 CTSC (0.46) CTSCKCNH2
SCHEMBL2892493 0.82 CTSC (0.63) CTSCKCNH2CTSK
SCHEMBL290293 0.80 CTSC (0.50) CTSCKCNH2CTSKBRD4
SCHEMBL290319 0.79 CTSC (0.42) CTSCKCNH2CTSK
SCHEMBL299100 0.78 CTSC (0.49) CTSCKCNH2
SCHEMBL290245 0.78 CTSS (0.39) CTSK
SCHEMBL289727 0.76 CTSC (0.54) CTSCCTSK
SCHEMBL290265 0.76 CTSC (0.34) CTSCKCNH2CTSK
SCHEMBL290665 0.76 CTSC (0.34) CTSCKCNH2CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed