SCHEMBL290245

SCHEMBL290245

COc1ccc(-c2ccc(CCN(C#N)C(=O)C3(NC(=O)O)CCOCC3)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
POLB P06746 3/20 0.39
MAPT P10636 2/20 0.38
FKBP1A P62942 1/20 0.38
CNR1 P21554 3/20 0.38
CNR2 P34972 3/20 0.38
HTR2A P28223 1/20 0.38
OPRK1 P41145 1/20 0.38
MMP1 P03956 1/20 0.38
MMP13 P45452 1/20 0.38
ALDH1A1 P00352 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALOX5 P09917 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL289589 0.85 RORC (0.37) MMP1MMP13
SCHEMBL290153 0.85 CD274 (0.35) CTSKMMP1MMP13
SCHEMBL290265 0.84 CTSC (0.34) CTSSCTSK
SCHEMBL290665 0.84 CTSC (0.34) CTSK
SCHEMBL289882 0.84 CTSC (0.32) CTSS
SCHEMBL290311 0.82 MMP12 (0.44) MMP13
SCHEMBL290431 0.81 GAA (0.48) POLBMAPTALDH1A1SMN1; SMN2
SCHEMBL290319 0.79 CTSC (0.42) CTSK
SCHEMBL288780 0.79 CTSC (0.40)
SCHEMBL290292 0.78 CTSC (0.47) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed