SCHEMBL289727

SCHEMBL289727

CN1C(=O)Cc2ccc(-c3ccc(CCN(C#N)C(=O)C4(NC(=O)O)CCOCC4)cc3)cc21

nearest known ligand 0.54

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CTSC P53634 20/20 0.54
CTSK P43235 7/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290319 0.81 CTSC (0.42) CTSCCTSK
SCHEMBL290265 0.81 CTSC (0.34) CTSCCTSK
SCHEMBL290665 0.81 CTSC (0.34) CTSCCTSK
SCHEMBL288985 0.80 MMP1 (0.41) CTSCCTSK
SCHEMBL290023 0.80 CTSC (0.45) CTSC
SCHEMBL2888765 0.80 CTSC (0.78) CTSCCTSK
SCHEMBL290245 0.79 CTSS (0.39) CTSK
SCHEMBL290311 0.79 MMP12 (0.44) CTSC
SCHEMBL289589 0.78 RORC (0.37) CTSC
SCHEMBL290109 0.78 CTSC (0.52) CTSCCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed