SCHEMBL29010808

SCHEMBL29010808

Cc1sccc1C1=NCCc2c(F)cccc21

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.34
GRM1 Q13255 1/20 0.34
NOS2 P35228 1/20 0.34
MAPK10 P53779 1/20 0.33
MAPK14 Q16539 1/20 0.33
CYP19A1 P11511 2/20 0.32
HTR1A P08908 2/20 0.32
HTR7 P34969 2/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
SRD5A1 P18405 1/20 0.31
TYMS P04818 1/20 0.31
MAOA P21397 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29010816 0.83 MAPK10 (0.38) GRM5GRM1NOS2MAPK10MAPK14
SCHEMBL29010834 0.76 NOS2 (0.46) NOS2MAPK10MAPK14HTR1AHTR7
SCHEMBL1009344 0.75 CYP19A1 (0.41) GRM5GRM1CYP19A1HTR1AHTR7
SCHEMBL28329716 0.69 ACHE (0.39)
SCHEMBL14246816 0.69 GABRA5 (0.32) MAPK10MAPK14
SCHEMBL3070384 0.69 NISCH (0.38) HTR1AHTR7CYP11B1CYP11B2
SCHEMBL29010811 0.68 MAPK10 (0.37) NOS2MAPK10MAPK14CYP19A1CYP11B2
SCHEMBL14246726 0.66 ALDH1A1 (0.39) MAPK10MAPK14MAOA
SCHEMBL29010851 0.66 MEN1 (0.42) NOS2MAPK10MAPK14TYMS
SCHEMBL6724928 0.65 MAPK10 (0.45) MAPK10MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116200357-B Imine reductase mutant and application thereof in synthesis of chiral tetrahydroisoquinoline 中国科学院天津工业生物技术研究所 2024-10-29 CN claimed
CN-116200357-A Imine reductase mutant and application thereof in synthesis of chiral tetrahydroisoquinoline 中国科学院天津工业生物技术研究所 2023-06-02 CN claimed
CN-116200357-B Imine reductase mutant and application thereof in synthesis of chiral tetrahydroisoquinoline 中国科学院天津工业生物技术研究所 2024-10-29 CN disclosed
CN-116200357-A Imine reductase mutant and application thereof in synthesis of chiral tetrahydroisoquinoline 中国科学院天津工业生物技术研究所 2023-06-02 CN disclosed