SCHEMBL29020110

SCHEMBL29020110

C[C@H](N)c1ccc(-c2ccc(O)cc2)c(F)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 5/20 0.64
CYP2C19 P33261 3/20 0.64
CYP2C9 P11712 2/20 0.64
CYP3A4 P08684 1/20 0.64
AKR1C3 P42330 6/20 0.49
AKR1C2 P52895 6/20 0.49
PTGS1 P23219 3/20 0.49
PTGS2 P35354 3/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
PSEN1 P49768 2/20 0.49
PSEN2 P49810 2/20 0.49
APH1B Q8WW43 2/20 0.49
NCSTN Q92542 2/20 0.49
APH1A Q96BI3 2/20 0.49
PSENEN Q9NZ42 2/20 0.49
FABP2 P12104 1/20 0.49
TSHR P16473 1/20 0.49
AKR1C4 P17516 1/20 0.49
ADRA2B P18089 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL765486 0.86 CYP2C19 (0.68) APPCYP2C19CYP2C9CYP3A4AKR1C3
SCHEMBL12327018 0.83 LMNA (0.64) CYP2C19CYP2C9AKR1C3AKR1C2PTGS1
4'-Hydroxyflurbiprofen SCHEMBL7040151 0.80 APP (0.97) APPCYP2C19CYP2C9CYP3A4AKR1C3
4'-Hydroxyflurbiprofen SCHEMBL6450842 0.80 APP (0.97) APPCYP2C19CYP2C9CYP3A4AKR1C3
SCHEMBL17524312 0.80 APP (0.81) APPCYP2C19CYP2C9CYP3A4AKR1C3
SCHEMBL2778899 0.78 APP (1.00) APPCYP2C19CYP2C9CYP3A4AKR1C3
SCHEMBL38659424 0.76 ESR1 (0.70) APPCYP2C19CYP2C9CYP3A4ESR1
SCHEMBL20497350 0.76 ESR1 (0.54) CYP2C19CYP2C9CYP3A4PTGS1DRD3
SCHEMBL18664389 0.76 ESR1 (0.54) CYP2C19CYP2C9CYP3A4PTGS1DRD3
SCHEMBL18664397 0.76 ESR1 (0.54) CYP2C19CYP2C9CYP3A4PTGS1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed