SCHEMBL29020124

SCHEMBL29020124

Nc1cc(-c2nc(C(=O)O)cc(-c3ccc(Cl)cc3)n2)ccn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 5/20 0.51
MCL1 Q07820 1/20 0.49
CTRC Q99895 3/20 0.48
MAP4K4 O95819 3/20 0.47
MKNK1 Q9BUB5 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46
GABRP O00591 1/20 0.44
GABRD O14764 1/20 0.44
GABRA1 P14867 1/20 0.44
GABRB1 P18505 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA2 P47869 1/20 0.44
GABRB2 P47870 1/20 0.44
GABRA4 P48169 1/20 0.44
GABRE P78334 1/20 0.44
GABRA6 Q16445 1/20 0.44
GABRG1 Q8N1C3 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29961695 1.00 KMO (0.51) KMOMCL1CTRCMAP4K4MKNK1
SCHEMBL29020201 0.85 KMO (0.51) KMOMCL1CTRCMAP4K4XDH
SCHEMBL29961689 0.85 KMO (0.51) KMOMCL1CTRCMAP4K4XDH
SCHEMBL21001267 0.83 MCL1 (0.61) KMOMCL1CTRCKDM4EMEN1
SCHEMBL29020197 0.82 MCL1 (0.55) KMOMCL1CTRCMAP4K4KDM4E
SCHEMBL29961681 0.79 KMO (0.56) KMOMCL1CTRCMAP4K4KDM4E
SCHEMBL29020139 0.79 KMO (0.56) KMOMCL1CTRCMAP4K4KDM4E
SCHEMBL1535621 0.78 CTRC (0.49) KMOMCL1CTRCMAP4K4GABRA2
SCHEMBL29808904 0.75 CTRC (0.55) KMOMCL1CTRCMKNK1MKNK2
SCHEMBL28803081 0.75 CTRC (0.55) KMOMCL1CTRCMKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed