SCHEMBL29020139

SCHEMBL29020139

O=C(O)c1cc(-c2ccc(Cl)cc2)nc(-c2cnc(Cl)nc2)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 4/20 0.56
MCL1 Q07820 2/20 0.53
CTRC Q99895 3/20 0.51
MAP4K4 O95819 3/20 0.48
ADORA3 P0DMS8 3/20 0.45
PTGES O14684 1/20 0.43
ALDH1A1 P00352 1/20 0.43
ALOX5 P09917 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
CASP7 P55210 1/20 0.43
HIF1A Q16665 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CA12 O43570 1/20 0.42
ALPL P05186 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29961681 1.00 KMO (0.56) KMOMCL1CTRCMAP4K4ADORA3
SCHEMBL21001267 0.88 MCL1 (0.61) KMOMCL1CTRCADORA3PTGES
SCHEMBL3408569 0.82 KMO (0.71) KMOMCL1CTRCPTGESALDH1A1
SCHEMBL29020197 0.81 MCL1 (0.55) KMOMCL1CTRCMAP4K4ADORA3
SCHEMBL25581810 0.81 MALT1 (0.47) ADORA3ALDH1A1ALPLKDM4E
SCHEMBL29020155 0.80 KMO (0.69) KMOMCL1CTRCPTGESALDH1A1
Potassium SCHEMBL29961618 0.80 KMO (0.69) KMOMCL1CTRCPTGESALDH1A1
SCHEMBL28803081 0.80 CTRC (0.55) KMOMCL1CTRCMEN1KMT2A
SCHEMBL29808904 0.80 CTRC (0.55) KMOMCL1CTRCMEN1KMT2A
SCHEMBL29020124 0.79 KMO (0.51) KMOMCL1CTRCMAP4K4ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed