SCHEMBL29020127

SCHEMBL29020127

CC(NC(=O)c1cc(-c2cnn(C)c2)nc(-c2cnn(C)c2)n1)c1cccc(F)c1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.49
PDPK1 O15530 1/20 0.47
RPS6KB1 P23443 1/20 0.47
LIPG Q9Y5X9 1/20 0.44
CLK1 P49759 2/20 0.43
PDE2A O00408 1/20 0.43
PFKFB3 Q16875 5/20 0.43
KCNT1 Q5JUK3 1/20 0.42
ROCK2 O75116 6/20 0.42
ROCK1 Q13464 3/20 0.42
RIPK1 Q13546 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29961598 1.00 MAPK1 (0.49) MAPK1PDPK1RPS6KB1LIPGCLK1
SCHEMBL29020122 1.00 MAPK1 (0.49) MAPK1PDPK1RPS6KB1LIPGCLK1
SCHEMBL29020217 0.93 CLK1 (0.47) MAPK1PDPK1RPS6KB1CLK1PDE2A
SCHEMBL29020220 0.93 CLK1 (0.47) MAPK1PDPK1RPS6KB1CLK1PDE2A
SCHEMBL29961633 0.93 CLK1 (0.47) MAPK1PDPK1RPS6KB1CLK1PDE2A
SCHEMBL29020117 0.85 KCNT1 (0.44) MAPK1CLK1KCNT1ROCK2ROCK1
SCHEMBL29020149 0.82 MAPK1 (0.44) MAPK1CLK1PDE2AKCNT1ROCK2
SCHEMBL29020185 0.82 ROCK2 (0.47) MAPK1CLK1PFKFB3KCNT1ROCK2
SCHEMBL29020159 0.81 CLK1 (0.50) MAPK1CLK1PDE2APFKFB3
SCHEMBL29961667 0.81 CLK1 (0.50) MAPK1CLK1PDE2APFKFB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed