SCHEMBL29020149

SCHEMBL29020149

CC(NC(=O)c1cc(-c2ccc(F)cc2)nc(-c2cnn(C)c2)n1)c1ccnc(F)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.44
ROCK2 O75116 4/20 0.43
PDE2A O00408 1/20 0.41
GPR55 Q9Y2T6 1/20 0.41
CLK1 P49759 4/20 0.41
PRKG1 Q13976 3/20 0.41
PRKACA P17612 2/20 0.41
PRKACG P22612 2/20 0.41
PRKACB P22694 2/20 0.41
AKT1 P31749 2/20 0.41
CYP2C9 P11712 1/20 0.41
ROCK1 Q13464 1/20 0.41
KIT P10721 3/20 0.40
KCNT1 Q5JUK3 1/20 0.40
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
JAK3 P52333 1/20 0.39
MKNK1 Q9BUB5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29020117 0.94 KCNT1 (0.44) MAPK1ROCK2CLK1PRKG1PRKACA
SCHEMBL29020210 0.93 CLK1 (0.48) MAPK1ROCK2CLK1PRKG1PRKACA
SCHEMBL29020185 0.93 ROCK2 (0.47) MAPK1ROCK2CLK1PRKG1PRKACA
SCHEMBL29020227 0.91 PDE2A (0.43) ROCK2PDE2APRKG1PRKACAPRKACG
SCHEMBL29020203 0.91 PHGDH (0.41) ROCK2CLK1PRKG1PRKACAPRKACG
SCHEMBL29020173 0.89 AHR (0.51) ROCK2PDE2ACLK1PRKG1PRKACA
SCHEMBL29020182 0.84 CLK1 (0.49) MAPK1ROCK2CLK1ROCK1KIT
SCHEMBL29020127 0.82 MAPK1 (0.49) MAPK1ROCK2PDE2ACLK1ROCK1
SCHEMBL29020122 0.82 MAPK1 (0.49) MAPK1ROCK2PDE2ACLK1ROCK1
SCHEMBL29961598 0.82 MAPK1 (0.49) MAPK1ROCK2PDE2ACLK1ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed