SCHEMBL29020117

SCHEMBL29020117

CC(NC(=O)c1cc(-c2cnn(C)c2)nc(-c2cnn(C)c2)n1)c1ccnc(F)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNT1 Q5JUK3 1/20 0.44
ROCK2 O75116 4/20 0.43
PRKG1 Q13976 3/20 0.42
PRKACA P17612 2/20 0.42
PRKACG P22612 2/20 0.42
PRKACB P22694 2/20 0.42
AKT1 P31749 2/20 0.42
MAPK1 P28482 5/20 0.41
CLK1 P49759 4/20 0.41
CYP2C9 P11712 1/20 0.41
ROCK1 Q13464 1/20 0.41
EGFR P00533 2/20 0.40
CLK2 P49760 1/20 0.40
LRRK2 Q5S007 1/20 0.40
RAB9A P51151 1/20 0.40
MET P08581 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29020185 0.96 ROCK2 (0.47) KCNT1ROCK2PRKG1PRKACAPRKACG
SCHEMBL29020149 0.94 MAPK1 (0.44) KCNT1ROCK2PRKG1PRKACAPRKACG
SCHEMBL29020210 0.93 CLK1 (0.48) KCNT1ROCK2PRKG1PRKACAPRKACG
SCHEMBL29020227 0.91 PDE2A (0.43) KCNT1ROCK2PRKG1PRKACAPRKACG
SCHEMBL29020203 0.91 PHGDH (0.41) ROCK2PRKG1PRKACAPRKACGPRKACB
SCHEMBL29020173 0.89 AHR (0.51) ROCK2PRKG1PRKACAPRKACGPRKACB
SCHEMBL29020127 0.85 MAPK1 (0.49) KCNT1ROCK2MAPK1CLK1ROCK1
SCHEMBL29961598 0.85 MAPK1 (0.49) KCNT1ROCK2MAPK1CLK1ROCK1
SCHEMBL29020122 0.85 MAPK1 (0.49) KCNT1ROCK2MAPK1CLK1ROCK1
SCHEMBL29020182 0.83 CLK1 (0.49) ROCK2MAPK1CLK1ROCK1CLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed