SCHEMBL29020173

SCHEMBL29020173

CC(NC(=O)c1cc(-c2ccc(OC(F)(F)F)cc2)nc(-c2cnn(C)c2)n1)c1ccnc(F)c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.51
PDE2A O00408 8/20 0.46
ABL1 P00519 3/20 0.45
BTK Q06187 1/20 0.43
ROCK2 O75116 3/20 0.42
ADORA3 P0DMS8 1/20 0.42
PRKG1 Q13976 2/20 0.41
CYP2C9 P11712 1/20 0.41
PRKACA P17612 1/20 0.41
PRKACG P22612 1/20 0.41
PRKACB P22694 1/20 0.41
AKT1 P31749 1/20 0.41
ROCK1 Q13464 1/20 0.41
BCR P11274 1/20 0.40
CLK1 P49759 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29020227 0.90 PDE2A (0.43) PDE2AROCK2PRKG1CYP2C9PRKACA
SCHEMBL29020149 0.89 MAPK1 (0.44) PDE2AROCK2PRKG1CYP2C9PRKACA
SCHEMBL29020117 0.89 KCNT1 (0.44) ROCK2PRKG1CYP2C9PRKACAPRKACG
SCHEMBL29020210 0.88 CLK1 (0.48) AHRROCK2PRKG1CYP2C9PRKACA
SCHEMBL29020185 0.87 ROCK2 (0.47) ROCK2PRKG1CYP2C9PRKACAPRKACG
SCHEMBL29020203 0.85 PHGDH (0.41) ROCK2PRKG1CYP2C9PRKACAPRKACG
SCHEMBL21004853 0.82 AHR (0.71) AHRPDE2AABL1BTKADORA3
SCHEMBL21004852 0.82 AHR (0.71) AHRPDE2AABL1BTKADORA3
SCHEMBL21001691 0.82 AHR (0.54) AHRPDE2AABL1BTKADORA3
SCHEMBL21001690 0.82 AHR (0.54) AHRPDE2AABL1BTKADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed