SCHEMBL29020178

SCHEMBL29020178

O=C(O)c1cc(-c2ccc(OC(F)(F)F)cc2)nc(Cl)n1.[KH]

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.57
KMO O15229 2/20 0.57
ADORA3 P0DMS8 1/20 0.48
AKR1C2 P52895 1/20 0.48
AKR1C1 Q04828 1/20 0.48
SCN10A Q9Y5Y9 3/20 0.46
AURKA O14965 1/20 0.45
TPX2 Q9ULW0 1/20 0.45
MARS1 P56192 1/20 0.44
SCN9A Q15858 2/20 0.44
MCL1 Q07820 2/20 0.44
SCN2A Q99250 1/20 0.43
PPARD Q03181 1/20 0.43
ACP1 P24666 1/20 0.43
CHRNA7 P36544 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21001335 0.99 KMO (0.58) DHODHKMOADORA3AKR1C2AKR1C1
Potassium SCHEMBL29961825 0.97 DHODH (0.57) DHODHKMOADORA3AKR1C2AKR1C1
Potassium Ion SCHEMBL29020198 0.86 DHODH (0.50) DHODHKMOADORA3AKR1C2AKR1C1
SCHEMBL24060792 0.85 KMO (0.52) DHODHKMOADORA3SCN10ASCN9A
SCHEMBL21001359 0.85 ADORA3 (0.61) DHODHKMOADORA3AKR1C2AKR1C1
SCHEMBL29020161 0.82 KMO (0.61) KMOADORA3MARS1MCL1
SCHEMBL29062398 0.82 KMO (0.68) DHODHKMOADORA3SCN9AMCL1
SCHEMBL3408828 0.81 KMO (0.62) KMOADORA3MARS1MCL1
SCHEMBL29020155 0.80 KMO (0.69) DHODHKMOMCL1
Potassium SCHEMBL29961608 0.80 KMO (0.61) KMOADORA3MARS1MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed