SCHEMBL290100

SCHEMBL290100

Cc1nc(-c2cc3ccccc3s2)sc1CC=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.40
ERN1 O75460 4/20 0.39
APP P05067 2/20 0.37
ADRB2 P07550 1/20 0.37
CYP19A1 P11511 1/20 0.36
CA1 P00915 2/20 0.36
CA9 Q16790 2/20 0.36
CA2 P00918 1/20 0.36
NQO1 P15559 1/20 0.36
NQO2 P16083 1/20 0.36
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
CA12 O43570 1/20 0.34
IKBKB O14920 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34
PRKDC P78527 1/20 0.34
PTGS1 P23219 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3822637 0.82 CYP2A6 (0.46) CYP2A6APPADRB2CYP19A1CA1
SCHEMBL851867 0.77 SMN1; SMN2 (0.51)
SCHEMBL288142 0.76 KDM4E (0.54)
SCHEMBL290239 0.75 CYP2A6 (0.42) CYP2A6ERN1APPADRB2CYP19A1
SCHEMBL280311 0.74 CYP2A6 (0.37) CYP2A6APPADRB2CYP19A1NQO1
SCHEMBL259711 0.74 PTGS1 (0.35) CYP2A6ERN1APPADRB2CYP19A1
SCHEMBL289881 0.72 SMN1; SMN2 (0.61) CA1CA9CA2CA12
SCHEMBL3828069 0.71 LMNA (0.51) APPJAK2JAK3IKBKB
SCHEMBL289322 0.70 CYP2A6 (0.48) CYP2A6
SCHEMBL289614 0.70 KDM4E (0.64) JAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed