SCHEMBL3828017

SCHEMBL3828017

Cc1ccc(-c2nc(C)c(CO)s2)s1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
MAPT P10636 2/20 0.37
NPC1 O15118 2/20 0.37
HSD17B10 Q99714 2/20 0.37
GFER P55789 1/20 0.37
KDM4E B2RXH2 5/20 0.35
SRC P12931 1/20 0.33
ZAP70 P43403 1/20 0.33
SYK P43405 1/20 0.33
GAA P10253 1/20 0.33
TP53 P04637 3/20 0.33
LMNA P02545 1/20 0.33
TRPV3 Q8NET8 1/20 0.33
HPGD P15428 1/20 0.33
NFKB1 P19838 1/20 0.33
RAB9A P51151 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PRMT6 Q96LA8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3822427 0.84 ALDH1A1 (0.42) ALDH1A1MAPTNPC1HSD17B10GFER
SCHEMBL13678345 0.82 MAPT (0.37) ALDH1A1MAPTNPC1HSD17B10GFER
Hydrochloric Acid SCHEMBL3826264 0.81 MAPT (0.36) ALDH1A1MAPTNPC1HSD17B10GFER
SCHEMBL289837 0.80 DPP4 (0.53) ALDH1A1MAPTNPC1HSD17B10KDM4E
SCHEMBL3436682 0.78 KDM4E (0.58) ALDH1A1MAPTNPC1HSD17B10KDM4E
SCHEMBL290239 0.77 CYP2A6 (0.42) LMNATRPV3
SCHEMBL8989130 0.75 KDM4E (0.54) MAPTKDM4EGAATP53LMNA
SCHEMBL3077683 0.75 SMN1; SMN2 (0.56) ALDH1A1MAPTNPC1KDM4EGAA
SCHEMBL17066355 0.75 ALDH1A1 (0.42) ALDH1A1MAPTNPC1HSD17B10GFER
SCHEMBL95917 0.72 RAB9A (0.56) ALDH1A1MAPTNPC1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2096111-A1 PYRAZOLES AND USE THEREOF AS DRUGS Japan Tobacco Inc. (JP) 2009-09-02 EP disclosed
US-20090036450-A1 PYRAZOLE COMPOUNDS AND USE THEREOF JAPAN TOBACCO, INC. (JP) 2009-02-05 US disclosed
US-20090036450-A1 PYRAZOLE COMPOUNDS AND USE THEREOF JAPAN TOBACCO, INC. (JP) 2009-02-05 US disclosed
US-20090036450-A1 PYRAZOLE COMPOUNDS AND USE THEREOF JAPAN TOBACCO, INC. (JP) 2009-02-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090036450-A1 PYRAZOLE COMPOUNDS AND USE THEREOF PYGL, GYS2, G6PC1 ALDH1A1 775/4885MAPT 2112/4885NPC1 2552/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.