SCHEMBL29024045

SCHEMBL29024045

CN1CC(CC2OCCO2)(c2ccccn2)CCC1=O

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.33
EPHX2 P34913 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
DRD2 P14416 4/20 0.33
DRD3 P35462 4/20 0.33
HSD11B1 P28845 2/20 0.32
SLC6A9 P48067 2/20 0.32
SIGMAR1 Q99720 1/20 0.32
OPRL1 P41146 1/20 0.32
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29024060 0.86 OPRM1 (0.34) OPRM1EPHX2CHRM2CHRM4CHRM5
SCHEMBL28270921 0.84 OPRM1 (0.35) OPRM1EPHX2CHRM2CHRM4CHRM5
SCHEMBL28270989 0.83 HSD11B1 (0.39) OPRM1EPHX2CHRM2CHRM4CHRM5
SCHEMBL28272495 0.80 GRIN1 (0.36) OPRM1EPHX2CHRM2CHRM4CHRM5
SCHEMBL28869101 0.78 CXCR3 (0.36) OPRM1EPHX2DRD2DRD3SLC6A2
SCHEMBL29967398 0.69 SLC6A2 (0.38) OPRM1EPHX2DRD2DRD3SLC6A2
SCHEMBL29968052 0.68 OPRM1 (0.57) OPRM1
SCHEMBL28270902 0.68 OPRM1 (0.57) OPRM1
SCHEMBL29024043 0.67 OPRM1 (0.37) OPRM1CHRM2CHRM4CHRM5CHRM1
Hydrochloric Acid SCHEMBL29968182 0.67 OPRM1 (0.56) OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109206417-B Opioid receptor agonists and uses thereof 四川海思科制药有限公司 2023-01-03 CN disclosed
CN-115124520-A Opioid receptor agonists and uses thereof 四川海思科制药有限公司 2022-09-30 CN disclosed