SCHEMBL29024481

SCHEMBL29024481

CC(C)COc1ccc(Cn2nc(CC3CC3)cc2C2CCN(C)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 19/20 0.42
ABCB11 O95342 1/20 0.40
CYP1A2 P05177 1/20 0.40
ADRB2 P07550 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD1 P21728 1/20 0.40
TBXA2R P21731 1/20 0.40
SLC6A2 P23975 1/20 0.40
HTR2C P28335 1/20 0.40
GPR183 P32249 1/20 0.40
CYP2C19 P33261 1/20 0.40
ADRA1A P35348 1/20 0.40
OPRM1 P35372 1/20 0.40
APLNR P35414 1/20 0.40
DRD3 P35462 1/20 0.40
CX3CR1 P49238 1/20 0.40
SLC6A3 Q01959 1/20 0.40
KCNH2 Q12809 1/20 0.40
GPR65 Q8IYL9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29024489 0.88 ABL1 (0.39) HTR2AABL1
SCHEMBL29024642 0.87 HTR2A (0.41) HTR2A
SCHEMBL29024647 0.86 HTR2A (0.51) HTR2AABCB11CYP1A2ADRB2CHRM2
SCHEMBL30478109 0.83 LTA4H (0.36) CYP1A2HRH3
SCHEMBL29024482 0.83 HTR2A (0.40) HTR2AABCB11CYP1A2ADRB2CHRM2
SCHEMBL30478119 0.78 SLC16A3 (0.38) HRH3
SCHEMBL29024639 0.75 SLC16A3 (0.41) HTR2AABL1
SCHEMBL29024635 0.73 TP53 (0.39) HTR2AHRH3
SCHEMBL29024637 0.73 HTR2A (0.47) HTR2AABCB11CYP1A2ADRB2CHRM2
SCHEMBL30478103 0.71 LTA4H (0.36) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116354925-A Pyrazole derivatives and use thereof 江苏恩华药业股份有限公司 2023-06-30 CN claimed
CN-116354925-A Pyrazole derivatives and use thereof 江苏恩华药业股份有限公司 2023-06-30 CN disclosed