SCHEMBL29025864

SCHEMBL29025864

CN(C)C=Nc1ccc(C2CCN(C(=O)OC(C)(C)C)CC2)cc1C#N

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.46
GPR119 Q8TDV5 14/20 0.43
NAMPT P43490 1/20 0.43
PDE4B Q07343 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
JAK3 P52333 2/20 0.40
LCK P06239 1/20 0.40
BTK Q06187 1/20 0.40
JAK2 O60674 1/20 0.39
PTK2 Q05397 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30126023 0.90 PDE4B (0.44) RETGPR119PDE4BMAPTJAK3
SCHEMBL30127474 0.90 PDE4B (0.44) RETGPR119PDE4BMAPTJAK3
SCHEMBL30126772 0.90 PDE4B (0.44) RETGPR119PDE4BMAPTJAK3
SCHEMBL29025845 0.86 QDPR (0.38) RET
SCHEMBL22076873 0.83 BTK (0.40) RETJAK3BTK
SCHEMBL25353312 0.82 ALDH1A1 (0.45) RETGPR119NAMPTMAPT
SCHEMBL30576110 0.82 ALDH1A1 (0.45) RETGPR119NAMPTMAPT
SCHEMBL30126320 0.82 ALDH1A1 (0.45) RETGPR119NAMPTMAPT
SCHEMBL30576111 0.82 ALDH1A1 (0.45) RETGPR119NAMPTMAPT
SCHEMBL30140211 0.81 GPR119 (0.49) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109422755-B Nitrogen-containing heterocyclic compound, preparation method, intermediate, composition and application 上海医药集团股份有限公司 2023-07-04 CN disclosed
CN-109422755-A A kind of nitrogen-containing heterocycle compound, preparation method, intermediate, composition and application 上海医药集团股份有限公司 2019-03-05 CN disclosed