SCHEMBL29026141

SCHEMBL29026141

COC(=O)c1ccc2nc(C(F)C(F)F)c(=O)[nH]c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.57
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
LMNA P02545 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
BRD4 O60885 1/20 0.49
PARP1 P09874 3/20 0.47
CSNK2A1 P68400 1/20 0.46
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
MMP8 P22894 1/20 0.46
MMP13 P45452 1/20 0.46
GRB7 Q14451 3/20 0.44
IRAK4 Q9NWZ3 1/20 0.43
NPY5R Q15761 2/20 0.42
MMP1 P03956 1/20 0.42
MMP3 P08254 1/20 0.42
MMP7 P09237 1/20 0.42
ADORA3 P0DMS8 1/20 0.41
PTGS1 P23219 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29397532 0.85 HTT (0.56) HTTKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL22963743 0.85 HTT (0.56) HTTKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL22963779 0.80 KDM4E (0.56) HTTKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL29396283 0.80 KDM4E (0.56) HTTKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL30908290 0.79 KDM4E (0.61) HTTKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL30349840 0.78 ALDH1A1 (0.64) HTTKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL6304842 0.78 KDM4E (0.70) HTTKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL22963740 0.77 HTT (0.59) HTTKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL29396281 0.77 HTT (0.59) HTTKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL22963739 0.77 HTT (0.65) HTTKDM4EALDH1A1LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116348115-A Combination of antibody-drug conjugate and PARP1 selective inhibitor 阿斯利康(英国)有限公司 2023-06-27 CN disclosed