SCHEMBL29131122

SCHEMBL29131122

COC(=O)c1c(CC#N)ccc(F)c1I

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 18/20 0.38
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29199348 0.83 BDKRB1 (0.38) BDKRB1CA12CA1CA2CA7
SCHEMBL29131126 0.82 CNR2 (0.40) BDKRB1CA12CA1CA2CA7
SCHEMBL2020273 0.81 BDKRB1 (0.37) BDKRB1CA12CA1CA2CA7
SCHEMBL29131091 0.81 BDKRB1 (0.38) BDKRB1
SCHEMBL29026652 0.79 BDKRB1 (0.47) BDKRB1CA12CA1CA2CA7
SCHEMBL29131129 0.79 SLC6A3 (0.35) BDKRB1ALDH1A1HSD17B10
SCHEMBL4203546 0.74 CA12 (0.44) CA12CA1CA2CA7CA9
SCHEMBL31401179 0.74 CA12 (0.44) CA12CA1CA2CA7CA9
SCHEMBL2334086 0.74 DPP4 (0.46) BDKRB1CA12CA1CA2CA7
SCHEMBL1867302 0.73 CA12 (0.41) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117903192-A Preparation method of 3-methoxy isoquinoline compound intermediate 上海相辉医药科技有限公司 2024-04-19 CN claimed
CN-117903192-A Preparation method of 3-methoxy isoquinoline compound intermediate 上海相辉医药科技有限公司 2024-04-19 CN disclosed
CN-117263959-A Preparation and application of aromatic KRAS mutant protein inhibitor 药雅科技(上海)有限公司 2023-12-22 CN disclosed