SCHEMBL29035532

SCHEMBL29035532

O=C(O)C(O)C(O)(C(=O)O)C1CCNCC1.O=C(O)c1n[nH]cc1NC(=O)c1c(Cl)cccc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 4/20 0.47
CDK5 Q00535 3/20 0.47
CDK4 P11802 2/20 0.47
CDK14 O94921 15/20 0.44
CCNY Q8ND76 15/20 0.44
CCNT1 O60563 2/20 0.44
CDK9 P50750 2/20 0.44
CDK5R1 Q15078 2/20 0.44
CCNA2 P20248 2/20 0.44
CCNA1 P78396 2/20 0.44
CASK O14936 1/20 0.44
CDKL5 O76039 1/20 0.44
CCNB2 O95067 1/20 0.44
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
MAK P20794 1/20 0.44
CDK11B P21127 1/20 0.44
CCND1 P24385 1/20 0.44
CCNE1 P24864 1/20 0.44
CCND3 P30281 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29035529 0.81 CDK14 (0.51) CDK2CDK5CDK4CDK14CCNY
SCHEMBL954955 0.78 KMT2A (0.51) CDK2CDK5CDK4CDK14CCNY
SCHEMBL8219606 0.75 TYK2 (0.52) CDK14CCNYMEN1KMT2A
At-7519 SCHEMBL955568 0.75 CDK5 (0.67) CDK2CDK5CDK4CDK14CCNY
SCHEMBL4488401 0.74 CDK14 (0.48) CDK2CDK5CDK4CDK14CCNY
At-7519 SCHEMBL31046986 0.74 CDK5 (0.66) CDK2CDK5CDK4CDK14CCNY
At-7519 SCHEMBL953647 0.74 CDK5 (0.66) CDK2CDK5CDK4CDK14CCNY
At-7519 SCHEMBL1069453 0.74 CDK5 (0.62) CDK2CDK5CDK4CDK14CCNY
SCHEMBL8261519 0.72 CDK5 (0.49) CDK2CDK5CDK4CDK14CCNY
SCHEMBL8044614 0.72 CDK5 (0.60) CDK2CDK5CDK4CDK14CCNY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109705090-B Tartaric acid addition salts of 3, 4-disubstituted 1H-pyrazole compounds and crystalline forms thereof 上海君实生物医药科技股份有限公司 2023-06-20 CN disclosed
CN-109705090-B Tartaric acid addition salts of 3, 4-disubstituted 1H-pyrazole compounds and crystalline forms thereof 上海君实生物医药科技股份有限公司 2023-06-20 CN disclosed