SCHEMBL29036003

SCHEMBL29036003

COC(=O)[C@H](N=C=O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.55
MEN1 O00255 2/20 0.42
ALDH1A1 P00352 2/20 0.42
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GAA P10253 1/20 0.39
SLC6A3 Q01959 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8853888 1.00 KMT2A (0.55) KMT2AMEN1ALDH1A1PTGS1PTGS2
SCHEMBL3578270 0.80 SRC (0.46) LMNACYP1A2CYP2D6MAPK1
SCHEMBL8627633 0.80 SRC (0.46) LMNACYP1A2CYP2D6MAPK1
SCHEMBL8508888 0.79 ALDH1A1 (0.50) KMT2AMEN1ALDH1A1LMNACYP1A2
SCHEMBL23515278 0.76 ALDH1A1 (0.40) KMT2AMEN1ALDH1A1TSHRHSD17B10
SCHEMBL16192842 0.75 MIF (0.36) KMT2AALDH1A1LMNACYP2D6MAPK1
SCHEMBL988808 0.75 HPGD (0.42) KMT2AALDH1A1LMNACYP2D6
SCHEMBL14521257 0.75 KMT2A (0.53) KMT2AMEN1ALDH1A1PTGS1PTGS2
SCHEMBL3909040 0.74 HPGD (0.37) ALDH1A1LMNAMAPK1
SCHEMBL2984292 0.73 KMT2A (0.51) KMT2AMEN1ALDH1A1PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232130-A APN and AKT double-target-point inhibitor and preparation method and application thereof 山东大学 2022-10-25 CN claimed
CN-115232130-B APN and AKT double-target inhibitor and preparation method and application thereof 山东大学 2024-01-12 CN disclosed
CN-115232130-A APN and AKT double-target-point inhibitor and preparation method and application thereof 山东大学 2022-10-25 CN disclosed