SCHEMBL290399

SCHEMBL290399

COc1ccc(-c2ccc(-c3nc(C)c(C(=O)O)s3)s2)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.48
SMN1; SMN2 Q16637 3/20 0.46
HSD17B1 P14061 1/20 0.46
HSD17B2 P37059 1/20 0.46
RAB9A P51151 3/20 0.45
GAA P10253 1/20 0.45
TARBP2 Q15633 1/20 0.45
ALPL P05186 1/20 0.44
KMT2A Q03164 4/20 0.44
POLB P06746 3/20 0.44
MEN1 O00255 3/20 0.44
XDH P47989 1/20 0.44
NPC1 O15118 3/20 0.43
ALDH1A1 P00352 2/20 0.43
RXFP1 Q9HBX9 2/20 0.43
CYP1A1 P04798 2/20 0.43
CYP1B1 Q16678 2/20 0.43
HPGD P15428 1/20 0.43
TP53 P04637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3435518 0.89 SMN1; SMN2 (0.51) KDM4ESMN1; SMN2RAB9AGAATARBP2
SCHEMBL288845 0.86 ALDH1A1 (0.54) KDM4ESMN1; SMN2HSD17B1HSD17B2RAB9A
SCHEMBL289862 0.85 APP (0.55) KDM4ESMN1; SMN2HSD17B1HSD17B2RAB9A
SCHEMBL289635 0.81 KDM4E (0.57) KDM4ESMN1; SMN2RAB9AGAATARBP2
SCHEMBL290387 0.80 KDM4E (0.47) KDM4ESMN1; SMN2RAB9AGAATARBP2
SCHEMBL289964 0.80 SMN1; SMN2 (0.57) KDM4ESMN1; SMN2HSD17B1HSD17B2RAB9A
SCHEMBL3435042 0.79 KDM4E (0.57) KDM4ESMN1; SMN2RAB9AGAATARBP2
SCHEMBL14800560 0.78 KDM4E (0.53) KDM4ESMN1; SMN2RAB9AGAATARBP2
SCHEMBL19523348 0.77 XDH (0.68) KDM4ERAB9AGAATARBP2XDH
SCHEMBL3436284 0.77 KDM4E (0.59) KDM4ESMN1; SMN2RAB9AGAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed