SCHEMBL29044477

SCHEMBL29044477

Cc1nc(Nc2cccnc2)sc1CC(=O)N(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 2/20 0.47
CDK5 Q00535 10/20 0.46
CDK5R1 Q15078 10/20 0.46
PIK3CA P42336 1/20 0.44
HPGD P15428 5/20 0.43
MAPT P10636 4/20 0.43
KDM4E B2RXH2 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
TRPV4 Q9HBA0 1/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
CDK2 P24941 1/20 0.42
GSK3B P49841 1/20 0.42
ALDH1A1 P00352 3/20 0.42
PPARG P37231 2/20 0.42
NCOA2 Q15596 2/20 0.42
NCOA1 Q15788 2/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30522192 1.00 PIK3CG (0.47) PIK3CGCDK5CDK5R1PIK3CAHPGD
SCHEMBL29044481 0.87 PTGDR2 (0.53) PIK3CGCDK5CDK5R1PIK3CAHPGD
SCHEMBL30522187 0.87 PTGDR2 (0.53) PIK3CGCDK5CDK5R1PIK3CAHPGD
SCHEMBL29044465 0.85 MAPT (0.50) PIK3CGCDK5CDK5R1PIK3CAHPGD
SCHEMBL29044470 0.79 MAPT (0.47) PIK3CGCDK5CDK5R1PIK3CAHPGD
SCHEMBL29044441 0.78 LMNA (0.58) CDK5CDK5R1MAPTKDM4ESMN1; SMN2
SCHEMBL11395592 0.77 CYP1A2 (0.56) HPGDMAPTKDM4ESMN1; SMN2ALDH1A1
SCHEMBL29044449 0.77 MAPT (0.47) PIK3CGCDK5CDK5R1PIK3CAHPGD
SCHEMBL30522185 0.77 MAPT (0.47) PIK3CGCDK5CDK5R1PIK3CAHPGD
SCHEMBL8738341 0.75 RAB9A (0.66) PIK3CGCDK5CDK5R1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116531373-A Thiazole compound, pharmaceutical composition and application thereof 上海日馨医药科技股份有限公司 2023-08-04 CN disclosed