SCHEMBL29045871

SCHEMBL29045871

CC(=O)N[C@H](C)c1nccc2c1[nH]c1c(Br)cccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 5/20 0.41
CDK9 P50750 4/20 0.41
DYRK1B Q9Y463 4/20 0.41
L3MBTL1 Q9Y468 6/20 0.40
ALOX12 P18054 5/20 0.40
DYRK2 Q92630 3/20 0.38
NPC1 O15118 3/20 0.37
RAB9A P51151 2/20 0.37
NCOA3 Q9Y6Q9 1/20 0.37
PARP14 Q460N5 1/20 0.37
OPRM1 P35372 1/20 0.37
PIM1 P11309 1/20 0.34
PIM3 Q86V86 1/20 0.34
ROCK2 O75116 2/20 0.34
DYRK3 O43781 1/20 0.34
ACACB O00763 1/20 0.34
ACACA Q13085 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29045875 1.00 DYRK1A (0.41) DYRK1ACDK9DYRK1BL3MBTL1ALOX12
SCHEMBL29985509 1.00 DYRK1A (0.41) DYRK1ACDK9DYRK1BL3MBTL1ALOX12
SCHEMBL29045947 0.86 L3MBTL1 (0.41) L3MBTL1ALOX12NPC1RAB9ANCOA3
SCHEMBL29986915 0.86 L3MBTL1 (0.41) L3MBTL1ALOX12NPC1RAB9ANCOA3
SCHEMBL29045950 0.86 L3MBTL1 (0.41) L3MBTL1ALOX12NPC1RAB9ANCOA3
SCHEMBL29045951 0.82 PARP14 (0.54) DYRK1AL3MBTL1NPC1RAB9APARP14
SCHEMBL29045946 0.82 PARP14 (0.54) DYRK1AL3MBTL1NPC1RAB9APARP14
SCHEMBL29045902 0.80 AR (0.42) DYRK1AL3MBTL1PARP14PIM1PIM3
SCHEMBL29045900 0.80 AR (0.42) DYRK1AL3MBTL1PARP14PIM1PIM3
SCHEMBL29986202 0.80 AR (0.42) DYRK1AL3MBTL1PARP14PIM1PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304597-B Beta-carboline compounds and application thereof in preparation of medicines for treating or preventing tumor diseases 中国科学院深圳先进技术研究院 2023-10-20 CN disclosed
CN-115304597-A Beta-carboline compounds and application thereof in preparing medicines for treating or preventing tumor diseases 中国科学院深圳先进技术研究院 2022-11-08 CN disclosed