SCHEMBL2904785

SCHEMBL2904785

O=C(/C=C/c1ccc(F)c(Cl)c1)N1CCC(=O)N(CCCN2CC(O)CCC2CO)CC1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 3/20 0.40
ITGB2 P05107 3/20 0.38
ICAM1 P05362 3/20 0.38
ITGAL P20701 3/20 0.38
GPR183 P32249 5/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
PYGL P06737 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2899153 0.92 CCR2 (0.39) CCR2ITGB2ICAM1ITGALGPR183
SCHEMBL2897127 0.91 CCR2 (0.45) CCR2ITGB2ICAM1ITGALGPR183
SCHEMBL2903670 0.89 ITGB2 (0.41) CCR2ITGB2ICAM1ITGALGPR183
SCHEMBL2905112 0.88 ITGB2 (0.38) CCR2ITGB2ICAM1ITGALGPR183
SCHEMBL2897251 0.87 ITGB2 (0.41) CCR2ITGB2ICAM1ITGALGPR183
SCHEMBL2904266 0.85 PYGL (0.42) CCR2ITGB2ICAM1ITGALGPR183
SCHEMBL2904263 0.85 PYGL (0.42) CCR2ITGB2ICAM1ITGALGPR183
SCHEMBL2904260 0.85 PYGL (0.42) CCR2ITGB2ICAM1ITGALGPR183
SCHEMBL2904597 0.85 CCR2 (0.44) CCR2ITGB2ICAM1ITGALGPR183
SCHEMBL2905016 0.84 CCR2 (0.47) CCR2ITGB2ICAM1ITGALGPR183

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed