SCHEMBL29050657

SCHEMBL29050657

CC(C)(O)NC(=O)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.61
CYP2C9 P11712 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
EPHX1 P07099 1/20 0.55
HDAC3 O15379 1/20 0.52
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
IDO1 P14902 1/20 0.52
ALOX15 P16050 1/20 0.52
HDAC1 Q13547 1/20 0.52
CA9 Q16790 1/20 0.52
HDAC7 Q8WUI4 1/20 0.52
HDAC2 Q92769 1/20 0.52
HSD17B10 Q99714 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
NCOR2 Q9Y618 1/20 0.52
GAA P10253 1/20 0.48
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL408310 0.84 CYP2C9 (0.67) POLBCYP2C9SMN1; SMN2EPHX1HDAC3
SCHEMBL10504078 0.83 POLB (0.58) POLBCYP2C9SMN1; SMN2EPHX1HDAC3
Fluoride SCHEMBL2310518 0.83 CYP2C9 (0.65) POLBCYP2C9SMN1; SMN2EPHX1HDAC3
SCHEMBL28820732 0.83 POLB (0.61) POLBCYP2C9SMN1; SMN2EPHX1HDAC3
Bromide SCHEMBL6851253 0.83 CYP2C9 (0.65) POLBCYP2C9SMN1; SMN2EPHX1HDAC3
Hydrochloric Acid SCHEMBL22076570 0.83 CYP2C9 (0.65) POLBCYP2C9SMN1; SMN2EPHX1HDAC3
SCHEMBL29201540 0.83 CYP2C9 (0.65) POLBCYP2C9SMN1; SMN2EPHX1HDAC3
SCHEMBL13416406 0.82 ALOX15 (0.56) POLBCYP2C9SMN1; SMN2EPHX1HDAC3
SCHEMBL9359968 0.82 POLB (0.56) POLBCYP2C9SMN1; SMN2EPHX1HDAC3
SCHEMBL343830 0.81 POLB (0.65) POLBCYP2C9SMN1; SMN2EPHX1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116589467-A Degradation of Bruton's Tyrosine Kinase (BTK) by conjugation of BTK inhibitors with E3 ligase ligands and methods of use thereof 百济神州有限公司 2023-08-15 CN disclosed
CN-116589466-A Degradation of Bruton's Tyrosine Kinase (BTK) by conjugation of BTK inhibitors with E3 ligase ligands and methods of use thereof 百济神州有限公司 2023-08-15 CN disclosed