Bromide

Bromide

SCHEMBL6851253

Br.CC(C)(C)NC(=O)c1ccccc1

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.65
SMN1; SMN2 Q16637 1/20 0.65
EPHX1 P07099 1/20 0.65
POLB P06746 2/20 0.61
HDAC3 O15379 1/20 0.52
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
IDO1 P14902 1/20 0.52
ALOX15 P16050 1/20 0.52
HDAC1 Q13547 1/20 0.52
CA9 Q16790 1/20 0.52
HDAC7 Q8WUI4 1/20 0.52
HDAC2 Q92769 1/20 0.52
HSD17B10 Q99714 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
NCOR2 Q9Y618 1/20 0.52
SIRT2 Q8IXJ6 1/20 0.50
GAA P10253 1/20 0.48
LMNA P02545 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL408310 0.98 CYP2C9 (0.67) CYP2C9SMN1; SMN2EPHX1POLBHDAC3
SCHEMBL29201540 0.96 CYP2C9 (0.65) CYP2C9SMN1; SMN2EPHX1POLBHDAC3
Fluoride SCHEMBL2310518 0.96 CYP2C9 (0.65) CYP2C9SMN1; SMN2EPHX1POLBHDAC3
Hydrochloric Acid SCHEMBL22076570 0.96 CYP2C9 (0.65) CYP2C9SMN1; SMN2EPHX1POLBHDAC3
Thiosulfuric Acid SCHEMBL11090482 0.87 CYP2C9 (0.56) CYP2C9SMN1; SMN2EPHX1POLBHDAC3
Thiosulfuric Acid SCHEMBL11090486 0.87 EPHX1 (0.60) CYP2C9SMN1; SMN2EPHX1POLBHDAC3
SCHEMBL17865779 0.86 LMNA (0.58) CYP2C9SMN1; SMN2EPHX1POLBHDAC1
SCHEMBL6416083 0.86 NPC1 (0.60) CYP2C9SMN1; SMN2EPHX1POLBGAA
SCHEMBL15946358 0.85 CACNA1B (0.67) SMN1; SMN2POLBLMNAHTTNPC1
SCHEMBL29050657 0.83 POLB (0.61) CYP2C9SMN1; SMN2EPHX1POLBHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1386912-A1 CYCLIC AMIDINE DERIVATIVE Eisai Co., Ltd. (JP) 2004-02-04 EP disclosed