SCHEMBL29051908

SCHEMBL29051908

CC(C)(CO[Si](c1ccccc1)(c1ccccc1)C(C)(C)C)N1CCc2ccc([N+](=O)[O-])cc2CC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 6/20 0.40
GRIN1 Q05586 2/20 0.38
DRD2 P14416 1/20 0.37
CPT2 P23786 1/20 0.36
CPT1A P50416 1/20 0.36
AKR1C3 P42330 2/20 0.36
SMYD2 Q9NRG4 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HPGD P15428 1/20 0.35
ADRA2A P08913 1/20 0.35
PNMT P11086 1/20 0.35
ABL1 P00519 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29051805 0.83 NR1H2 (0.37) GRIN2BGRIN1DRD2SMYD2
SCHEMBL30468501 0.76 PNMT (0.43) GRIN2BGRIN1DRD2AKR1C3HPGD
SCHEMBL30468430 0.71 GRIN1 (0.39) GRIN2BGRIN1DRD2SMYD2MEN1
SCHEMBL28693868 0.70 MEN1 (0.37) MEN1KMT2AHPGDABL1
SCHEMBL29052165 0.69 DRD2 (0.46) DRD2AKR1C3ADRA2APNMT
SCHEMBL6622197 0.69 PPARD (0.46) MEN1KMT2A
SCHEMBL30878905 0.69 ALDH1A1 (0.46) MEN1KMT2A
SCHEMBL5574184 0.68 IDO1 (0.50) AKR1C3MEN1KMT2A
SCHEMBL1950525 0.68 PNMT (0.54) GRIN2BMEN1KMT2AHPGDADRA2A
SCHEMBL22559463 0.68 HTR6 (0.43) MEN1KMT2AABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116332910-A 2-aminopyrimidine derivatives as kinase inhibitors, preparation and use thereof 江苏威凯尔医药科技有限公司 2023-06-27 CN disclosed