SCHEMBL29059448

SCHEMBL29059448

O=C(O)[C@@H](CC1(C(F)(F)F)CC1)NCCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GGT1 P19440 1/20 0.43
CYP2C19 P33261 3/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP1A2 P05177 1/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
MLYCD O95822 2/20 0.39
EPHX1 P07099 1/20 0.39
TSHR P16473 1/20 0.38
SIGMAR1 Q99720 2/20 0.37
ACE P12821 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
PLAAT3 P53816 1/20 0.37
PLAAT5 Q96KN8 1/20 0.37
PLAAT2 Q9NWW9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29059381 0.80 CYP1A2 (0.39) CYP2C19CYP3A4CYP2D6CYP2C9CYP1A2
SCHEMBL29059374 0.80 GGT1 (0.46) GGT1CYP2C19CYP3A4CYP2D6CYP2C9
SCHEMBL24298217 0.74 ALDH1A1 (0.40) GGT1ACE
SCHEMBL24298266 0.74 MEN1 (0.42) KMT2AMEN1
SCHEMBL25362932 0.74 MEN1 (0.42) KMT2AMEN1
SCHEMBL7469306 0.74 GGT1 (0.54) GGT1CYP2C19CYP3A4CYP2D6CYP2C9
SCHEMBL7469320 0.74 GGT1 (0.54) GGT1CYP2C19CYP3A4CYP2D6CYP2C9
SCHEMBL27699637 0.74 MME (0.56) GGT1KMT2ASIGMAR1ACE
SCHEMBL8609013 0.74 GGT1 (0.54) GGT1CYP2C19CYP3A4CYP2D6CYP2C9
SCHEMBL27699635 0.74 MME (0.56) GGT1KMT2ASIGMAR1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116783204-A Modulators of cystic fibrosis transmembrane conductance regulator 弗特克斯药品有限公司 2023-09-19 CN disclosed
CN-116601158-A Modulators of cystic fibrosis transmembrane conductance regulator 弗特克斯药品有限公司 2023-08-15 CN disclosed