SCHEMBL29062256

SCHEMBL29062256

Cc1cccc(C(=O)NC2CCOC2)c1C

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.54
TAS1R1 Q7RTX1 1/20 0.54
TAS1R2 Q8TE23 1/20 0.54
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.49
GLA P06280 1/20 0.45
PTGES O14684 1/20 0.44
FASN P49327 1/20 0.43
NAMPT P43490 2/20 0.43
P2RX7 Q99572 2/20 0.42
POLB P06746 1/20 0.41
HPGDS O60760 1/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CHRM4 P08173 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20477095 0.92 SMN1; SMN2 (0.57) TAS1R3TAS1R1TAS1R2NPC1RAB9A
SCHEMBL13162643 0.89 NPC1 (0.64) NPC1RAB9ASMN1; SMN2GLAFASN
SCHEMBL13634628 0.89 NPC1 (0.64) NPC1RAB9ASMN1; SMN2GLAFASN
SCHEMBL1987660 0.84 TAS1R3 (0.64) TAS1R3TAS1R1TAS1R2NPC1RAB9A
SCHEMBL13162693 0.80 NPC1 (0.72) NPC1RAB9ASMN1; SMN2GLAPOLB
SCHEMBL27204928 0.79 CNR2 (0.49) NPC1RAB9ASMN1; SMN2NAMPTHPGDS
SCHEMBL27171970 0.79 CNR2 (0.49) NPC1RAB9ASMN1; SMN2NAMPTHPGDS
SCHEMBL14688259 0.78 TAS1R3 (0.62) TAS1R3TAS1R1TAS1R2NPC1RAB9A
SCHEMBL28503120 0.77 P2RX7 (0.47) TAS1R3TAS1R1TAS1R2NPC1RAB9A
SCHEMBL28949389 0.77 CRBN (0.48) NPC1RAB9ASMN1; SMN2NAMPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117069728-A PI4KIII beta inhibitors 葛兰素史克知识产权开发有限公司 2023-11-17 CN claimed
CN-111868063-B PI4KIII beta inhibitors 葛兰素史克知识产权开发有限公司 2023-08-01 CN claimed
CN-117069728-A PI4KIII beta inhibitors 葛兰素史克知识产权开发有限公司 2023-11-17 CN disclosed