SCHEMBL2906852

SCHEMBL2906852

FC(F)Oc1ccc(I)nc1OCC1CC1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 15/20 0.43
PDE4D Q08499 12/20 0.43
PDE4A P27815 6/20 0.43
PDE4C Q08493 6/20 0.43
ABCB11 O95342 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30350527 0.81 FFAR4 (0.43) PDE4BPDE4DPDE4APDE4C
SCHEMBL2909751 0.81 FFAR4 (0.43) PDE4BPDE4DPDE4APDE4C
SCHEMBL4148746 0.79 MEN1 (0.36) PDE4BPDE4DPDE4APDE4C
SCHEMBL2907667 0.77 FPR2 (0.34) PDE4BPDE4DPDE4APDE4C
SCHEMBL2905855 0.75 PDE4D (0.39) PDE4BPDE4DPDE4APDE4C
SCHEMBL23982177 0.74 PDE4D (0.56) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL30476643 0.74 PDE4D (0.56) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL2908835 0.73 PDE4B (0.35) PDE4BPDE4DPDE4APDE4C
SCHEMBL2907660 0.72 TRPM8 (0.33)
SCHEMBL2418124 0.71 APP (0.47) PDE4BPDE4DPDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1692109-B1 PHOSPHODIESTERASE 4 INHIBITORS, INCLUDING N-SUBSTITUTED DIARYLAMINE ANALOGS MEMORY PHARM CORP (US) 2010-08-18 EP disclosed
US-20090118270-A1 PHOSPHODIESTERASE 4 INHIBITORS TALAMAS FRANCISCO XAVIER 2009-05-07 US disclosed
US-20070049611-A1 Phosphodiesterase 4 inhibitors F. HOFFMANN-LA ROCHE AG (CH) 2007-03-01 US disclosed
US-20050222207-A1 Phosphodiesterase 4 inhibitors, including N-substituted diarylamine analogs MEMORY PHARMACEUTICAL CORPORATION 2005-10-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070049611-A1 Phosphodiesterase 4 inhibitors PDE4A, PDE3B, PDE4B PDE4B 3/4885PDE4D 6/4885PDE4A 1/4885
US-20050222207-A1 Phosphodiesterase 4 inhibitors, including N-substituted diarylamine analogs PDE4A, PDE4B, PDE3B PDE4B 2/4885PDE4D 6/4885PDE4A 1/4885
US-20090118270-A1 PHOSPHODIESTERASE 4 INHIBITORS PDE4A, PDE3B, PDE4B PDE4B 3/4885PDE4D 6/4885PDE4A 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.