SCHEMBL2907419

SCHEMBL2907419

COC(=O)c1cccc(-c2c(C)cc(N)nc2C)c1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 3/20 0.47
KLKB1 P03952 1/20 0.41
ALDH1A1 P00352 6/20 0.41
CFTR P13569 1/20 0.41
HSD17B10 Q99714 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
MAPK10 P53779 2/20 0.40
MEN1 O00255 2/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
GAA P10253 2/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
PTK2B Q14289 1/20 0.39
NCOA1 Q15788 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2898209 0.80 MYC (0.54) ALDH1A1CFTRHSD17B10SLC6A2SLC6A4
SCHEMBL1707844 0.78 CYP3A4 (0.45) ALDH1A1CFTRHSD17B10SLC6A2SLC6A4
SCHEMBL13139655 0.77 REN (0.58) REN
SCHEMBL13117379 0.77 ATR (0.40) ALDH1A1HSD17B10SLC6A2SLC6A4SLC6A3
SCHEMBL13117454 0.76 KDM4E (0.38) RENALDH1A1HSD17B10SLC6A2SLC6A4
SCHEMBL28675430 0.76 PDCD1 (0.50) ALDH1A1CFTRHSD17B10SLC6A2SLC6A4
SCHEMBL13117458 0.76 KDM4E (0.35) ALDH1A1SLC6A2SLC6A4SLC6A3MAPK10
SCHEMBL13117455 0.76 KDM4E (0.35) ALDH1A1SLC6A2SLC6A4SLC6A3MAPK10
SCHEMBL29634134 0.75 TSHR (0.53) ALDH1A1CFTRHSD17B10SLC6A2SLC6A4
SCHEMBL19849652 0.75 TSHR (0.53) ALDH1A1CFTRHSD17B10SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100267775-A1 OXADIAZOLIDINEDIONE COMPOUND ASTELLAS PHARMA INC. (JP) 2010-10-21 US disclosed
US-20100267775-A1 OXADIAZOLIDINEDIONE COMPOUND ASTELLAS PHARMA INC. (JP) 2010-10-21 US disclosed
EP-2216330-A1 OXADIAZOLIDINEDIONE COMPOUND Astellas Pharma Inc. (JP) 2010-08-11 EP disclosed
EP-2216330-A1 OXADIAZOLIDINEDIONE COMPOUND Astellas Pharma Inc. (JP) 2010-08-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100267775-A1 OXADIAZOLIDINEDIONE COMPOUND GPR119, GLP1R, GPR4 REN 1017/4885KLKB1 2052/4885ALDH1A1 2370/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.