SCHEMBL2907649

SCHEMBL2907649

CCc1cc(NC(=O)CC(C)=O)ccc1NC(=O)CC(C)=O

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.55
KMT2A Q03164 4/20 0.55
ALDH1A1 P00352 3/20 0.55
KDM4E B2RXH2 2/20 0.55
CYP1A2 P05177 1/20 0.55
CYP2C19 P33261 1/20 0.55
HIF1A Q16665 1/20 0.55
POLB P06746 4/20 0.50
MAPT P10636 2/20 0.50
TSHR P16473 1/20 0.50
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA4 P22748 1/20 0.47
CA7 P43166 1/20 0.47
NR4A1 P22736 1/20 0.42
RAB9A P51151 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2913783 0.81 POLB (0.61) MEN1KMT2AALDH1A1KDM4ECYP1A2
SCHEMBL2913865 0.80 MEN1 (0.61) MEN1KMT2AALDH1A1KDM4ECYP1A2
SCHEMBL2904641 0.80 KMT2A (0.55) MEN1KMT2AALDH1A1KDM4ECYP1A2
SCHEMBL5368510 0.80 KMT2A (0.55) MEN1KMT2AALDH1A1KDM4ECYP1A2
SCHEMBL2908421 0.78 KDM4E (0.51) MEN1KMT2AALDH1A1KDM4ECYP1A2
SCHEMBL593172 0.78 MAPT (0.74) MEN1KMT2AALDH1A1KDM4ECYP1A2
SCHEMBL2914555 0.78 MEN1 (0.66) MEN1KMT2AALDH1A1KDM4ECYP1A2
SCHEMBL8752424 0.77 HDAC3 (0.61) MEN1KMT2AALDH1A1POLBMAPT
SCHEMBL31570103 0.77 HDAC3 (0.61) MEN1KMT2AALDH1A1POLBMAPT
SCHEMBL10704337 0.76 ALDH1A1 (0.51) MEN1KMT2AALDH1A1KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6756486-B1 LAKED DISAZO YELLOW PIGMENTS HAVING DESIRABLE GREEN SHADE, HEAT STABILITY, GOOD STRENGTH, BLEED RESISTANCE, MIGRATION RESISTANCE, AND LOW OR NO TOXICITY ENGELHARD CORPORATION 2004-06-29 US claimed
EP-1668080-B1 NON-MIGRATING MEALLIZED DISAZO GREEN SHADE YELLOW PIGMENT ENGELHARD CORP (US) 2010-08-11 EP disclosed
EP-1668080-A1 NON-MIGRATING MEALLIZED DISAZO GREEN SHADE YELLOW PIGMENT Engelhard Corporation (US) 2006-06-14 EP disclosed
WO-2005033212-A1 NON-MIGRATING MEALLIZED DISAZO GREEN SHADE YELLOW PIGMENT ENGELHARD CORPORATION (US) 2005-04-14 WO disclosed
US-6756486-B1 LAKED DISAZO YELLOW PIGMENTS HAVING DESIRABLE GREEN SHADE, HEAT STABILITY, GOOD STRENGTH, BLEED RESISTANCE, MIGRATION RESISTANCE, AND LOW OR NO TOXICITY ENGELHARD CORPORATION 2004-06-29 US disclosed
EP-1104444-B1 STRONG GREEN-SHADE YELLOW DISAZO PIGMENT ENGELHARD CORP (US) 2002-12-18 EP disclosed
US-6254671-B1 Very green-shade yellow metallized disazo pigment ENGELHARD CORPORATION 2001-07-03 US disclosed
EP-1104444-A1 STRONG GREEN-SHADE YELLOW DISAZO PIGMENT Engelhard Corporation (US) 2001-06-06 EP disclosed
WO-2001036540-A1 VERY GREEN-SHADE YELLOW METALLIZED DISAZO PIGMENT ENGELHARD CORPORATION (US) 2001-05-25 WO disclosed
WO-2000009614-A1 STRONG GREEN-SHADE YELLOW DISAZO PIGMENT ENGELHARD CORPORATION (US) 2000-02-24 WO disclosed
US-5889162-A COUPLING A DIAZONIUM COMPONENT MADE FROM ONE OR MORE AROMATIC AMINES SUCH AS 2-ETHOXYANILINE WITH AT LEAST ONE COUPLING AGENT; SUITABLE FOR USE IN PLASTICS, PAINTS AND INKS ENGELHARD CORPORATION (US) 1999-03-30 US disclosed
EP-0025164-B1 DISAZO COMPOUNDS, PROCESS FOR THEIR PREPARATION AND USE HOECHST AKTIENGESELLSCHAFT (DE) 1983-04-13 EP disclosed
EP-0025164-A1 Disazo compounds, process for their preparation and use HOECHST AKTIENGESELLSCHAFT (DE) 1981-03-18 EP disclosed