SCHEMBL29076894

SCHEMBL29076894

COC(=O)c1cc(C)nc(C)c1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.51
HPGD P15428 3/20 0.51
ALDH1A1 P00352 3/20 0.51
L3MBTL1 Q9Y468 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
KMT2A Q03164 2/20 0.45
GAA P10253 1/20 0.44
BACE1 P56817 1/20 0.43
MEN1 O00255 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
HSD17B10 Q99714 2/20 0.41
SPR P35270 1/20 0.41
MAPT P10636 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
CASP3 P42574 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23884915 0.83 NQO2 (0.47) KDM4EHPGDALDH1A1L3MBTL1GAA
SCHEMBL27151963 0.81 KDM4E (0.47) KDM4EHPGDALDH1A1GAAHSD17B10
SCHEMBL31310191 0.81 KDM4E (0.56) KDM4EHPGDALDH1A1L3MBTL1TDP1
SCHEMBL31310092 0.81 KDM4E (0.49) KDM4EHPGDALDH1A1L3MBTL1TDP1
SCHEMBL30823904 0.81 KDM4E (0.47) KDM4EHPGDALDH1A1GAAHSD17B10
SCHEMBL13590587 0.78 ALDH1A1 (0.45) KDM4EHPGDALDH1A1TDP1KMT2A
SCHEMBL4174949 0.75 SMN1; SMN2 (0.58) KDM4EHPGDALDH1A1L3MBTL1KMT2A
SCHEMBL28478763 0.74 NPSR1 (0.50) KDM4EHPGDALDH1A1L3MBTL1TDP1
SCHEMBL12500156 0.74 NPC1 (0.57) KDM4EHPGDALDH1A1L3MBTL1TDP1
SCHEMBL31310214 0.73 KDM4E (0.42) KDM4EHPGDALDH1A1L3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114907318-B Isonicotinic acid-pyrazole derivative and preparation method and application thereof 郑州大学 2023-08-11 CN disclosed
CN-114907318-A Isonicotinic acid-pyrazole derivative and preparation method and application thereof 郑州大学 2022-08-16 CN disclosed