SCHEMBL29077465

SCHEMBL29077465

N#Cc1cc2c(cn1)CCN(C(=O)O)C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
TAS1R2 Q8TE23 1/20 0.38
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
ALDH1A1 P00352 3/20 0.36
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
THRB P10828 1/20 0.34
S1PR1 P21453 2/20 0.34
MAPK1 P28482 2/20 0.34
GAA P10253 1/20 0.34
KDM4E B2RXH2 1/20 0.33
USP2 O75604 1/20 0.33
PKM P14618 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25428617 0.81 NR1H2 (0.55) MAPTMAPK1ESR2
SCHEMBL27940431 0.78 HPGD (0.47) ALDH1A1SMN1; SMN2MAPK1GAAHPGD
SCHEMBL2594044 0.78 NOS3 (0.47) MAPTKMT2AMEN1NPC1TP53
SCHEMBL22466192 0.78 GAA (0.39) KMT2AMEN1ALDH1A1SMN1; SMN2GAA
SCHEMBL5600099 0.77 KMT2A (0.45) MAPTTAS1R3TAS1R1TAS1R2KMT2A
SCHEMBL28707742 0.77 CYP11B2 (0.39) ALDH1A1
SCHEMBL25209956 0.76 GPR142 (0.59) MAPTKMT2AMEN1ALDH1A1NPC1
SCHEMBL22583571 0.75 CYP11B2 (0.38) ALDH1A1KDM4EHPGD
SCHEMBL29077472 0.74 KMT2A (0.34) KMT2AMEN1NPC1SMN1; SMN2MAPK1
SCHEMBL28369820 0.74 AKR1C3 (0.52) MAPTESR1ESR2SPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116783190-A N- (phenylaminocarbonyl) tetrahydroisoquinolines and related compounds as modulators of GPR65 帕蒂奥斯治疗有限公司 2023-09-19 CN disclosed