SCHEMBL29078409

SCHEMBL29078409

COc1ccc(NS(=O)(=O)CCN2CCN(c3ncccn3)CC2)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.47
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA7 P43166 2/20 0.45
DRD2 P14416 3/20 0.44
MYD88 Q99836 1/20 0.43
KDM4E B2RXH2 2/20 0.42
POLB P06746 1/20 0.42
HTT P42858 2/20 0.41
NPC1 O15118 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HTR1A P08908 2/20 0.41
DRD3 P35462 2/20 0.41
DRD1 P21728 1/20 0.41
HTR2A P28223 1/20 0.41
ABCB1 P08183 1/20 0.41
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SLC22A12 Q96S37 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30585260 0.83 TSHR (0.53) TSHRMYD88KDM4EPOLBHTT
SCHEMBL29078383 0.80 MYD88 (0.51) DRD2MYD88POLBHTTNPC1
SCHEMBL30585253 0.80 TSHR (0.47) TSHRMYD88POLBHTTNPC1
SCHEMBL29078361 0.76 MYD88 (0.55) TSHRMYD88POLBHTTNPC1
SCHEMBL29078402 0.76 ALDH1A1 (0.62) TSHRDRD2KDM4EPOLBHTT
SCHEMBL29078406 0.76 MYD88 (0.68) TSHRMYD88KDM4EPOLBHTT
SCHEMBL30585247 0.75 HTR7 (0.46) CA1CA2CA7POLBNPC1
SCHEMBL29078377 0.75 HTR7 (0.46) CA1CA2CA7POLBNPC1
SCHEMBL19303544 0.72 TSHR (0.63) TSHRKDM4EPOLBHTTNPC1
SCHEMBL29078379 0.70 KMT2A (0.54) CA1CA2CA7DRD2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116803981-A Piperazine-containing amide or sulfonamide anti-inflammatory compound and preparation method and application thereof 温州医科大学 2023-09-26 CN claimed
CN-116803981-A Piperazine-containing amide or sulfonamide anti-inflammatory compound and preparation method and application thereof 温州医科大学 2023-09-26 CN disclosed