SCHEMBL30585253

SCHEMBL30585253

COc1ccc(CN2CCN(CCS(=O)(=O)Nc3ccc(OC)nc3)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
ALDH1A1 P00352 2/20 0.46
LMNA P02545 2/20 0.46
NPC1 O15118 1/20 0.46
S1PR2 O95136 1/20 0.46
S1PR4 O95977 1/20 0.46
MAPT P10636 1/20 0.46
S1PR1 P21453 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TLR9 Q9NR96 1/20 0.46
SIGMAR1 Q99720 1/20 0.44
MYD88 Q99836 1/20 0.44
FAAH O00519 1/20 0.44
ACHE P22303 1/20 0.44
POLB P06746 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30585260 0.91 TSHR (0.53) TSHRALDH1A1LMNANPC1S1PR2
SCHEMBL29078361 0.87 MYD88 (0.55) TSHRALDH1A1LMNANPC1HTT
SCHEMBL29078406 0.81 MYD88 (0.68) TSHRALDH1A1LMNAMAPTHTT
SCHEMBL29078409 0.80 TSHR (0.47) TSHRALDH1A1LMNANPC1HTT
SCHEMBL29078375 0.79 CHKA (0.50) ALDH1A1LMNANPC1SIGMAR1FAAH
SCHEMBL30585266 0.79 CHKA (0.50) ALDH1A1LMNANPC1SIGMAR1FAAH
SCHEMBL29078372 0.77 ALDH1A1 (0.61) ALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL30585261 0.77 ALDH1A1 (0.61) ALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL29078383 0.75 MYD88 (0.51) ALDH1A1LMNANPC1MAPTHTT
SCHEMBL29078393 0.73 ACHE (0.53) ALDH1A1LMNAKMT2ASIGMAR1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116803981-A Piperazine-containing amide or sulfonamide anti-inflammatory compound and preparation method and application thereof 温州医科大学 2023-09-26 CN claimed
CN-116803981-A Piperazine-containing amide or sulfonamide anti-inflammatory compound and preparation method and application thereof 温州医科大学 2023-09-26 CN disclosed