SCHEMBL29078361

SCHEMBL29078361

COc1ccc(NS(=O)(=O)CCN2CCN(Cc3ccc([N+](=O)[O-])cc3)CC2)cn1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MYD88 Q99836 1/20 0.55
MEN1 O00255 2/20 0.47
PABPC1 P11940 2/20 0.47
KMT2A Q03164 2/20 0.47
POLB P06746 1/20 0.47
SMN1; SMN2 Q16637 4/20 0.46
HTT P42858 2/20 0.46
LMNA P02545 2/20 0.46
KCNJ1 P48048 2/20 0.44
KCNH2 Q12809 2/20 0.44
ALDH1A1 P00352 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
GAA P10253 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TSHR P16473 1/20 0.43
FAAH O00519 1/20 0.42
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29078406 0.90 MYD88 (0.68) MYD88MEN1PABPC1KMT2APOLB
SCHEMBL29078383 0.89 MYD88 (0.51) MYD88MEN1PABPC1KMT2APOLB
SCHEMBL30585253 0.87 TSHR (0.47) MYD88KMT2APOLBSMN1; SMN2HTT
SCHEMBL30585260 0.86 TSHR (0.53) MYD88MEN1PABPC1KMT2APOLB
SCHEMBL28954891 0.79 MYD88 (0.85) MYD88MEN1PABPC1KMT2ASMN1; SMN2
SCHEMBL29078394 0.79 MEN1 (0.60) MYD88MEN1PABPC1KMT2APOLB
SCHEMBL29078409 0.76 TSHR (0.47) MYD88MEN1KMT2APOLBSMN1; SMN2
SCHEMBL29078367 0.76 CHKA (0.47) SMN1; SMN2HTTLMNAALDH1A1GAA
SCHEMBL30585249 0.76 CHKA (0.47) SMN1; SMN2HTTLMNAALDH1A1GAA
SCHEMBL30585285 0.74 ALDH1A1 (0.46) MYD88SMN1; SMN2HTTLMNAKCNJ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116803981-A Piperazine-containing amide or sulfonamide anti-inflammatory compound and preparation method and application thereof 温州医科大学 2023-09-26 CN claimed
CN-116803981-A Piperazine-containing amide or sulfonamide anti-inflammatory compound and preparation method and application thereof 温州医科大学 2023-09-26 CN disclosed