SCHEMBL29085366

SCHEMBL29085366

Nc1nccc(C2CC2)c1Br

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.36
NOS3 P29474 4/20 0.33
NOS2 P35228 4/20 0.33
NOS1 P29475 2/20 0.33
CYP17A1 P05093 4/20 0.31
F12 P00748 1/20 0.31
PLAU P00749 1/20 0.31
NCF1 P14598 1/20 0.31
BACE1 P56817 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
GRIN3B O60391 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2C Q14957 1/20 0.31
PRKCI P41743 1/20 0.31
PDK2 Q15119 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29526095 0.79 NOS3 (0.45) RETNOS3NOS2NOS1CYP17A1
SCHEMBL928999 0.79 NOS3 (0.45) RETNOS3NOS2NOS1CYP17A1
SCHEMBL31240930 0.76 CYP17A1 (0.36) NOS3NOS2NOS1CYP17A1F12
SCHEMBL3668400 0.76 NOS2 (0.52) RETNOS3NOS2NOS1CYP17A1
SCHEMBL29864311 0.76 CYP17A1 (0.33) CYP17A1HTR2AHTR2CHTR2BPDK2
SCHEMBL30731660 0.73 KDM4E (0.41)
SCHEMBL27039119 0.73 KDM4E (0.41)
SCHEMBL22493647 0.72 USP7 (0.35) RETNOS3NOS2NOS1F12
SCHEMBL31312603 0.72 CYP17A1 (0.37) NOS3NOS2NOS1CYP17A1HTR2C
SCHEMBL28284231 0.72 TDO2 (0.40) NOS3NOS2NOS1CYP17A1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116867781-A Imidazo [1,2-a ] pyridine derivatives as IRAK4 inhibitors and their use in the treatment of diseases 渤健马萨诸塞州股份有限公司 2023-10-10 CN disclosed