SCHEMBL2909840

SCHEMBL2909840

N#Cc1ccc(NCCCn2cc(C(=O)O)c(-c3ccc(Cl)cc3Cl)c2)nc1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 5/20 0.55
TMPRSS4 Q9NRS4 1/20 0.46
CCNB2 O95067 1/20 0.44
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
RPS6KB1 P23443 1/20 0.44
CDK2 P24941 1/20 0.44
GSK3A P49840 1/20 0.44
LIMK1 P53667 1/20 0.44
TAOK1 Q7L7X3 1/20 0.44
CCNB3 Q8WWL7 1/20 0.44
SLK Q9H2G2 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
CSNK1G1 Q9HCP0 1/20 0.44
DPP7 Q9UHL4 2/20 0.42
IDH1 O75874 1/20 0.39
DPP4 P27487 9/20 0.39
DPP8 Q6V1X1 1/20 0.36
CCR6 P51684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2908173 0.88 GSK3B (0.47) GSK3BTMPRSS4CCNB2CDK1CCNB1
SCHEMBL2911030 0.86 GSK3B (0.46) GSK3BTMPRSS4CCNB2CDK1CCNB1
SCHEMBL2912712 0.86 GSK3B (0.46) GSK3BTMPRSS4CCNB2CDK1CCNB1
SCHEMBL2911764 0.86 GSK3B (0.46) GSK3BTMPRSS4CCNB2CDK1CCNB1
SCHEMBL2911861 0.86 GSK3B (0.46) GSK3BTMPRSS4CCNB2CDK1CCNB1
SCHEMBL2912436 0.84 F10 (0.41) GSK3B
SCHEMBL2911621 0.83 GSK3B (0.47) GSK3BTMPRSS4CCNB2CDK1CCNB1
SCHEMBL2912974 0.83 GSK3B (0.47) GSK3BCDK2DPP4
SCHEMBL1219415 0.75 GSK3B (0.51) GSK3BCCNB2CDK1CCNB1CDK2
SCHEMBL2909829 0.73 HCRTR1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed