SCHEMBL2911027

SCHEMBL2911027

COC1CCC(N2CCOCC2)Cc2c1cccc2[N+](=O)[O-]

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAPT P10636 8/20 0.38
ALDH1A1 P00352 3/20 0.38
LMNA P02545 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PKM P14618 1/20 0.37
MAPK1 P28482 2/20 0.36
KMT2A Q03164 2/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MEN1 O00255 1/20 0.36
CYP2C9 P11712 1/20 0.36
CTSB P07858 1/20 0.36
TDP1 Q9NUW8 2/20 0.36
POLB P06746 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2910804 0.79 ALDH1A1 (0.43) MAPTALDH1A1LMNASMN1; SMN2PKM
SCHEMBL2915008 0.75 SIGMAR1 (0.42) MAPTMAPK1TDP1
SCHEMBL2061689 0.72 SIGMAR1 (0.42) MAPTALDH1A1LMNAPKMMAPK1
SCHEMBL2062474 0.72 SIGMAR1 (0.42) MAPTALDH1A1LMNAPKMMAPK1
SCHEMBL3435490 0.70 CTSB (0.52) CYP1A2MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL2061632 0.70 ALK (0.42) MAPTALDH1A1LMNASMN1; SMN2KMT2A
SCHEMBL2908344 0.69 GAA (0.38) MAPTSMN1; SMN2GAA
SCHEMBL16571285 0.68 MEN1 (0.42) ALDH1A1LMNASMN1; SMN2KMT2AGAA
SCHEMBL2061311 0.67 ALK (0.42) CYP1A2CYP2C19MAPTALDH1A1LMNA
SCHEMBL2482410 0.65 ALDH1A1 (0.36) MAPTALDH1A1LMNASMN1; SMN2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222647-A1 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS Cephalon, Inc. (US) 2010-09-01 EP disclosed
WO-2008051547-A1 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS CEPHALON, INC. (US) 2008-05-02 WO disclosed