SCHEMBL29115489

SCHEMBL29115489

CNC(=O)c1cc(F)c(N2CCNCC2)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
HPGD P15428 4/20 0.48
KDM4E B2RXH2 3/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 1/20 0.48
CASP1 P29466 1/20 0.48
CYP2C19 P33261 1/20 0.48
ACLY P53396 1/20 0.44
LMNA P02545 4/20 0.44
HTT P42858 2/20 0.44
TSHR P16473 2/20 0.42
HSD17B10 Q99714 2/20 0.42
BRD4 O60885 1/20 0.42
CYP2J2 P51589 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MAPKAPK2 P49137 1/20 0.41
MAPT P10636 2/20 0.40
POLB P06746 1/20 0.40
APEX1 P27695 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29115675 0.88 ALDH1A1 (0.45) ALDH1A1HPGDKDM4ECYP1A2ACLY
SCHEMBL21832673 0.85 ALDH1A1 (0.45) ALDH1A1HPGDKDM4ECYP1A2ACLY
SCHEMBL27747368 0.77 MAPT (0.47) ALDH1A1HPGDKDM4ECYP1A2CYP3A4
SCHEMBL29115378 0.76 ACLY (0.39) ALDH1A1ACLYMAPKAPK2MAPK8MAPK9
SCHEMBL29115477 0.76 ADRB1 (0.56) CYP1A2CYP3A4CYP2C19HTTMAPT
SCHEMBL30542902 0.76 MAPT (0.50) ALDH1A1HPGDLMNATSHRNPSR1
SCHEMBL21360370 0.76 KDR (0.45) ALDH1A1HTR1A
SCHEMBL531792 0.76 MAPT (0.50) ALDH1A1HPGDLMNATSHRNPSR1
Hydrochloric Acid SCHEMBL31032930 0.75 MAPT (0.49) ALDH1A1HPGDLMNATSHRNPSR1
Hydrochloric Acid SCHEMBL30858323 0.75 MAPT (0.49) ALDH1A1HPGDLMNATSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116710433-A Selective PARP1 inhibitor and application thereof 成都百裕制药股份有限公司 2023-09-05 CN disclosed
WO-2022222966-A1 SELECTIVE PARP1 INHIBITOR AND APPLICATION THEREOF 成都百裕制药股份有限公司 2022-10-27 WO disclosed