SCHEMBL29124653

SCHEMBL29124653

CC(c1ccc(F)cc1)c1nc2cc(Br)cnc2[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
CDK5 Q00535 3/20 0.36
EGFR P00533 3/20 0.36
ABL1 P00519 2/20 0.36
RET P07949 2/20 0.36
KDR P35968 2/20 0.36
CDK7 P50613 2/20 0.36
PRKAA1 Q13131 2/20 0.36
AURKB Q96GD4 2/20 0.36
CLK4 Q9HAZ1 2/20 0.36
GSK3A P49840 2/20 0.36
GSK3B P49841 2/20 0.36
NTRK1 P04629 2/20 0.36
AURKA O14965 1/20 0.36
JAK2 O60674 1/20 0.36
PAK4 O96013 1/20 0.36
LCK P06239 1/20 0.36
FYN P06241 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14770635 0.85 DYRK1B (0.38) CDK5ABL1RETCDK7PRKAA1
SCHEMBL12309248 0.78 LMNA (0.40) CDK5ABL1RETKDRCDK7
SCHEMBL14770631 0.77 GSK3A (0.36) CDK5EGFRABL1RETCDK7
SCHEMBL14770525 0.77 APP (0.42)
SCHEMBL855351 0.76 CYP1A2 (0.43) CDK5ABL1RETKDRCDK7
SCHEMBL13620301 0.75 ALPL (0.37) CDK5EGFRABL1RETKDR
SCHEMBL14770524 0.74 APP (0.40)
SCHEMBL13607851 0.73 ALDH1A1 (0.47) CDK5ABL1RETKDRCDK7
SCHEMBL14770725 0.71 MEN1 (0.39) CDK5ABL1RETCDK7PRKAA1
SCHEMBL13607786 0.70 HPGD (0.44) CDK5ABL1RETKDRCDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116768889-A Novel CDK9 kinase inhibitor and preparation method and application thereof 厦门大学 2023-09-19 CN disclosed