SCHEMBL2912906

SCHEMBL2912906

CC(C)(C)c1cc(/C=C/c2ccc(NS(C)(=O)=O)cc2)cc(N2C(=O)CCNC2=O)c1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.39
TRPV1 Q8NER1 7/20 0.38
NR3C2 P08235 1/20 0.33
HDAC1 Q13547 1/20 0.33
EPHX2 P34913 1/20 0.32
NR1H4 Q96RI1 1/20 0.32
PIP4K2A P48426 1/20 0.32
PIP4K2B P78356 1/20 0.32
HDAC8 Q9BY41 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2913880 0.83 CYP3A4 (0.56) CYP3A4TRPV1
SCHEMBL2913728 0.83 CYP3A4 (0.56) CYP3A4TRPV1
SCHEMBL2908324 0.83 TRPV1 (0.39) CYP3A4TRPV1EPHX2NR1H4
SCHEMBL2910649 0.83 TDP2 (0.33) TRPV1NR3C2EPHX2NR1H4
SCHEMBL2111740 0.82 CYP3A4 (0.39) CYP3A4TRPV1NR3C2HDAC1EPHX2
SCHEMBL2111743 0.82 CYP3A4 (0.39) CYP3A4TRPV1NR3C2HDAC1EPHX2
SCHEMBL2909890 0.81 CA1 (0.42) TRPV1EPHX2NR1H4
SCHEMBL2912524 0.81 RAB9A (0.44) TRPV1EPHX2NR1H4
SCHEMBL2111741 0.80 CYP3A4 (0.39) CYP3A4TRPV1NR3C2HDAC1EPHX2
SCHEMBL1530141 0.78 TRPV1 (0.42) CYP3A4TRPV1NR3C2HDAC1PIP4K2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222646-A1 URACIL OR THYMINE DERIVATIVE FOR TREATING HEPATITIS C Abbott Laboratories (US) 2010-09-01 EP disclosed
EP-2203430-A1 N-PHENYL-DIOXO-HYDROPYRIMIDINES USEFUL AS HEPATITIS C VIRUS (HCV) INHIBITORS Abbott Laboratories (US) 2010-07-07 EP disclosed
WO-2009039135-A1 N-PHENYL-DIOXO-HYDROPYRIMIDINES USEFUL AS HEPATITIS C VIRUS (HCV) INHIBITORS ABBOTT LABORATORIES (US) 2009-03-26 WO disclosed
WO-2009039127-A1 URACIL OR THYMINE DERIVATIVE FOR TREATING HEPATITIS C ABBOTT LABORATORIES (US) 2009-03-26 WO disclosed