SCHEMBL29131091

SCHEMBL29131091

COC(=O)c1c(CC#N)ccc(F)c1C(C)C

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 17/20 0.38
GCGR P47871 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29131122 0.81 BDKRB1 (0.38) BDKRB1
SCHEMBL29199348 0.81 BDKRB1 (0.38) BDKRB1MEN1KMT2A
SCHEMBL29131126 0.80 CNR2 (0.40) BDKRB1
SCHEMBL29026652 0.77 BDKRB1 (0.47) BDKRB1MEN1KMT2A
SCHEMBL29131129 0.76 SLC6A3 (0.35) BDKRB1MEN1KMT2A
SCHEMBL10299409 0.72 CNR2 (0.38) BDKRB1MEN1KMT2A
SCHEMBL2334086 0.71 DPP4 (0.46) BDKRB1MEN1KMT2A
SCHEMBL4203546 0.71 CA12 (0.44) MEN1KMT2A
SCHEMBL31401179 0.71 CA12 (0.44) MEN1KMT2A
SCHEMBL14660758 0.70 KDM4E (0.40) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117903192-A Preparation method of 3-methoxy isoquinoline compound intermediate 上海相辉医药科技有限公司 2024-04-19 CN claimed
CN-117903192-A Preparation method of 3-methoxy isoquinoline compound intermediate 上海相辉医药科技有限公司 2024-04-19 CN disclosed
CN-117263959-A Preparation and application of aromatic KRAS mutant protein inhibitor 药雅科技(上海)有限公司 2023-12-22 CN disclosed