SCHEMBL29131129

SCHEMBL29131129

COC(=O)c1c(CC#N)ccc(F)c1C1CC1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 3/20 0.35
BDKRB1 P46663 12/20 0.35
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
SLC6A4 P31645 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HCRTR2 O43614 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29131122 0.79 BDKRB1 (0.38) BDKRB1ALDH1A1HSD17B10
SCHEMBL29199348 0.79 BDKRB1 (0.38) BDKRB1HPGDMEN1KMT2A
SCHEMBL29131126 0.77 CNR2 (0.40) BDKRB1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL29131091 0.76 BDKRB1 (0.38) BDKRB1MEN1KMT2A
SCHEMBL29026652 0.75 BDKRB1 (0.47) BDKRB1MEN1KMT2A
SCHEMBL27841029 0.71 ALDH1A1 (0.40) SLC6A3ALDH1A1HPGDTSHRHSD17B10
SCHEMBL31401179 0.70 CA12 (0.44) ALDH1A1HPGDTSHRHSD17B10MEN1
SCHEMBL4203546 0.70 CA12 (0.44) ALDH1A1HPGDTSHRHSD17B10MEN1
SCHEMBL2334086 0.70 DPP4 (0.46) BDKRB1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL28313 0.69 KDM4E (0.39) SLC6A3ALDH1A1HPGDTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117903192-A Preparation method of 3-methoxy isoquinoline compound intermediate 上海相辉医药科技有限公司 2024-04-19 CN claimed
CN-117903192-A Preparation method of 3-methoxy isoquinoline compound intermediate 上海相辉医药科技有限公司 2024-04-19 CN disclosed
CN-117263959-A Preparation and application of aromatic KRAS mutant protein inhibitor 药雅科技(上海)有限公司 2023-12-22 CN disclosed