SCHEMBL2913177

SCHEMBL2913177

NC(=O)C1(C(c2ccccc2)C(F)(F)F)CCCCC1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1C1 Q04828 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
HDAC4 P56524 2/20 0.33
GAA P10253 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
OPRK1 P41145 1/20 0.33
TSHR P16473 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL517632 0.76 ALOX5 (0.41) AKR1C1KMT2AALDH1A1OPRK1CYP1A2
SCHEMBL29985406 0.76 ALDH1A1 (0.32) AKR1C1KMT2AGAAALDH1A1OPRK1
SCHEMBL6942516 0.76 SLC6A2 (0.42) OPRK1
SCHEMBL5815457 0.73 CHRM2 (0.40) KMT2AMEN1ALDH1A1TSHRCYP2D6
SCHEMBL6472115 0.72 MME (0.37) KMT2AMEN1OPRK1
SCHEMBL516114 0.72 SRC (0.41) AKR1C1CYP1A2CYP2D6
SCHEMBL516716 0.72 LMNA (0.37) CYP1A2CYP2D6
SCHEMBL18342994 0.71 ALDH1A1 (0.40) KMT2AALDH1A1TSHRCYP2D6
SCHEMBL30816986 0.70 CNR2 (0.39) KMT2AMEN1ALDH1A1OPRK1CYP1A2
SCHEMBL30851542 0.70 CNR2 (0.39) KMT2AMEN1ALDH1A1OPRK1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2214487-A1 NOVEL SEH INHIBITORS AND THEIR USE GlaxoSmithKline LLC (US) 2010-08-11 EP disclosed
WO-2009049157-A1 NOVEL SEH INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO disclosed