SCHEMBL29132492

SCHEMBL29132492

C=CCOC(=O)NS(=O)(=O)N(CC(=O)OC(C)(C)C)c1c(OCc2ccccc2)cc2c(c1F)C[C@H](N(CCCC)C(=O)OCc1ccccc1)CC2

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 3/20 0.33
TMEM97 Q5BJF2 2/20 0.32
TRPM8 Q7Z2W7 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HTR2A P28223 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29626302 1.00 CCR5 (0.33) CCR5TMEM97TRPM8L3MBTL1HTR2A
SCHEMBL25338987 0.93 CCR5 (0.35) CCR5TMEM97TRPM8HTR2A
SCHEMBL29626474 0.85 CA1 (0.41) L3MBTL1
SCHEMBL29024337 0.85 CA1 (0.41) L3MBTL1
SCHEMBL29626395 0.85 CA1 (0.38) L3MBTL1
SCHEMBL29626309 0.84 ACACB (0.33)
SCHEMBL25339147 0.81 CA1 (0.39) L3MBTL1
SCHEMBL25194894 0.80 L3MBTL1 (0.31) L3MBTL1
SCHEMBL25339103 0.80 ACACB (0.33)
SCHEMBL29024310 0.80 GABRP (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116829555-A Protein tyrosine phosphatase inhibitors and methods of use thereof 卡里科生命科学有限责任公司 2023-09-29 CN disclosed