SCHEMBL29132996

SCHEMBL29132996

COCc1cc(-c2nnc(C3CN(C(=O)OC(C)(C)C)C3C(C)(C)C)o2)ccc1Br

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 2/20 0.37
TLR7 Q9NYK1 2/20 0.37
TSHR P16473 5/20 0.34
MAPT P10636 4/20 0.34
LMNA P02545 4/20 0.34
KMT2A Q03164 3/20 0.34
NPSR1 Q6W5P4 2/20 0.34
MEN1 O00255 2/20 0.34
HTT P42858 1/20 0.34
GPR119 Q8TDV5 1/20 0.33
ALDH1A1 P00352 4/20 0.33
SMN1; SMN2 Q16637 3/20 0.32
GAA P10253 1/20 0.32
THRB P10828 1/20 0.32
TLR9 Q9NR96 1/20 0.31
HDAC6 Q9UBN7 2/20 0.31
S1PR4 O95977 1/20 0.31
S1PR1 P21453 1/20 0.31
S1PR5 Q9H228 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29132973 0.75 ALDH1A1 (0.38) TLR8TLR7MAPTLMNAALDH1A1
SCHEMBL29133055 0.73 ALDH1A1 (0.52) TLR8TLR7MAPTALDH1A1TLR9
SCHEMBL29133064 0.67 NOTUM (0.43) TSHRMAPTLMNAKMT2AHTT
SCHEMBL29133160 0.67 SMN1; SMN2 (0.41) TLR8TLR7MAPTLMNAKMT2A
SCHEMBL29133017 0.66 DGAT1 (0.50) TLR8TLR7MAPTLMNAKMT2A
SCHEMBL12098306 0.65 KMT2A (0.61) TSHRMAPTLMNAKMT2ANPSR1
SCHEMBL12098303 0.65 KMT2A (0.61) TSHRMAPTLMNAKMT2ANPSR1
SCHEMBL30622248 0.65 KDM4E (0.49) MAPTLMNAKMT2ANPSR1MEN1
SCHEMBL15099854 0.64 ALDH1A1 (0.50) TLR8TLR7TSHRMAPTLMNA
SCHEMBL22602035 0.63 ALDH1A1 (0.54) TSHRMAPTLMNAKMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed